Code:
Serine/threonine protein kinase 12 AZD1152 DCL000452 Myeloid Leukemia Phase I/II
Serine/threonine protein kinase 12 AZD1152 DCL000452 Acute Myeloid Leukemia, Haematological malignancies Phase II
Serine/threonine protein kinase 12 MK-5108 DCL000572 Cancer; Neoplasms; Tumors Phase I
Serine/threonine protein kinase 12 TAK-901 DCL000657 Advanced malignancies Phase I
Serine/threonine protein kinase 12 AT-9283 DCL001068 Adult solid tumours, NHL, AML, ALL, CML, MDS and myelofibrosis Phase I/II
Serine/threonine protein kinase 12 CYC-116 DCL001070 Advanced solid tumours Terminated in Phase I
Serine/threonine protein kinase 12 GSK1070916 DCL001072 Advanced solid tumours Phase I
Serine/threonine protein kinase 12 PF-03814735 DCL001076 Advanced solid tumours Phase I
Serine/threonine protein kinase 12 PHA-739358 DCL001078 CML that relapsed after imatinib or BCR¨CABL-targeted therapy; Metastatic Hormone Refractory Prostate Cancer (MHRPC) Phase II
Serine/threonine protein kinase 12 VX-689 DCL001083 Cancer; Neoplasms; Tumors Phase I
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform SF1126 DCL000228 Solid Tumors Phase I
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform TG100-115 DCL000246 Angioedema, Myocardial infarction Phase I/II
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform XL147 DCL000262 Endometrial Cancer Phase II
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform XL765 DCL000264 Solid tumours; non-small-cell lung cancer; malignant gliomas Phase I/II
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform AZD6482 DCL000476 Thrombosis Phase II
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform LY294002 DCL000600 Cancer Discontinued in Phase I
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform PI3K alpha DCL000601 Cancer Discontinued in Phase I
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform BEZ235 DCL001085 Advanced solid tumours; Advanced breast cancer Phase I/II
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform BGT226 DCL001086 Solid tumours; Advanced breast cancer; Cowden¡¯s syndrome Phase I/II
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform BKM120 DCL001087 Metastatic Breast Cancer Phase I/II
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform GDC0941 DCL001088 Advanced solid tumours; non-Hodgkin¡¯s lymphoma Phase I
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform GSK1059615 DCL001089 Advanced solid tumours; metastatic breast cancer; endometrial cancer; lymphoma Terminated in Phase I
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform PX-866 DCL001090 Advanced solid tumours Phase I
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform CAL-101 DCL001091 Chronic lymphocytic leukaemia; acute myeloid leukaemia; non-Hodgkin¡¯s lymphoma Phase I
Phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit, gamma isoform GDC-0980 DCL001189 Advanced solid tumours, non-Hodgkin's lymphoma Phase I
Hexokinase D Lonidamine DCL000153 Benign Prostatic Hyperplasia, Prostate Disorders Terminated in Phase III
Hexokinase D PSN-101 DCL000201 Diabetes Mellitus Type 1 and 2 Phase I
Hexokinase D AZD1656 DCL000457 Type 2 Diabetes Mellitus Phase II
Hexokinase D AZD6370 DCL000475 Type 2 Diabetes Phase I completed
Hexokinase D R7201 DCL000614 Type 2 diabetes Phase II
Hexokinase D AZD5658 DCL001154 Obesity, Diabetes Phase I
mRNA of Clusterin OGX-011 DCL000186 Prostate Cancer, Breast Cancer, Lung Cancer Phase III
Kinesin-like protein KIF11 ARRY-520 DCL000053 Cancer/Tumors Phase I
Kinesin-like protein KIF11 Ispinesib DCL000139 Pediatric Phase I
Kinesin-like protein KIF11 Ispinesib DCL000139 Head and Neck Cancer, Renal Cell Carcinoma, Ovarian Cancer, Solid Tumors Phase II
Kinesin-like protein KIF11 Ispinesib DCL000139 Lung Cancer Phase II completed
Kinesin-like protein KIF11 SB-743921 DCL000224 Non-Hodgkin's Lymphoma, Cancer/Tumors Phase I/II
Kinesin-like protein KIF11 4SC-205 DCL001129 Solid tumour and malignant lymphoma Phase I
Neurotensin receptor type 1 CGX-1160 DCL000084 Acute or Chronic Pain Phase I completed
Neurotensin receptor type 1 Meclinertant DCL000163 Colorectal Cancer, Prostate Cancer, Schizophrenia, Schizoaffective Disorders, Psychosis, Depression, Lung Cancer Discontinued in Phase III
Ribosomal protein S6 kinase XL418 DCL000009 Solid Tumors Suspended in Phase I
Interstitial collagenase BMS 275291 DCL000003 Non-small Cell Lung Cancer, Hormone-refractory Prostate Cancer, Kaposi's Sarcoma Discontinued in Phase III
Interstitial collagenase Prinomastat DCL000004 Brain Cancer Discontinued in Phase III
Interstitial collagenase Prinomastat DCL000004 Lung Cancer, Prostate Cancer Trial halted
Interstitial collagenase Marimastat DCL000005 Pancreatic Cancer, Lung Cancer Discontinued in Phase III
Interstitial collagenase BB-3644 DCL000014 Cancer/Tumors Discontinued in Phase I
Interstitial collagenase XL784 DCL001039 Diabetic nephropathy Discontinued in Phase II
Interstitial collagenase Batimastat DPR000163 Cancers Discontinued in Phase I
Integrin beta